Files
rdkit/Code/GraphMol/Subgraphs/SubgraphUtils.cpp
Greg Landrum e2521dccbc add murcko decomposition;
be sure pathToSubmol copies over coordinates
2011-02-21 06:43:53 +00:00

238 lines
8.9 KiB
C++

// $Id$
//
// Copyright (C) 2003-2010 Greg Landrum and Rational Discovery LLC
//
// @@ All Rights Reserved @@
// This file is part of the RDKit.
// The contents are covered by the terms of the BSD license
// which is included in the file license.txt, found at the root
// of the RDKit source tree.
//
#include "SubgraphUtils.h"
#include "Subgraphs.h"
#include <RDGeneral/utils.h>
#include <GraphMol/RDKitBase.h>
#include <GraphMol/QueryAtom.h>
#include <GraphMol/QueryBond.h>
#include <iostream>
#include <algorithm>
#include <map>
#include <boost/tuple/tuple_comparison.hpp>
#include <RDGeneral/hash/hash.hpp>
namespace RDKit {
namespace Subgraphs {
ROMol *pathToSubmol(const ROMol &mol, const PATH_TYPE &path,
bool useQuery) {
INT_MAP_INT aIdxMap;
return pathToSubmol(mol, path, useQuery, aIdxMap);
}
ROMol *pathToSubmol(const ROMol &mol, const PATH_TYPE &path,
bool useQuery,
INT_MAP_INT &atomIdxMap) {
RWMol *subMol=new RWMol();
PATH_TYPE::const_iterator pathIter;
atomIdxMap.clear();
if (useQuery) {
// have to do this in two different blocks because of issues with variable scopes.
for(pathIter=path.begin(); pathIter!=path.end(); ++pathIter){
QueryBond *bond;
bond = new QueryBond(*(mol.getBondWithIdx(*pathIter)));
int begIdx=bond->getBeginAtomIdx();
int endIdx=bond->getEndAtomIdx();
if(atomIdxMap.find(begIdx)==atomIdxMap.end()){
QueryAtom *atom = new QueryAtom(*(mol.getAtomWithIdx(begIdx)));
int newAtomIdx=subMol->addAtom(atom,false,true);
atomIdxMap[begIdx] = newAtomIdx;
}
begIdx = atomIdxMap.find(begIdx)->second;
if(atomIdxMap.find(endIdx)==atomIdxMap.end()){
QueryAtom *atom = new QueryAtom(*(mol.getAtomWithIdx(endIdx)));
int newAtomIdx=subMol->addAtom(atom,false,true);
atomIdxMap[endIdx] = newAtomIdx;
}
endIdx = atomIdxMap.find(endIdx)->second;
bond->setOwningMol(subMol);
bond->setBeginAtomIdx(begIdx);
bond->setEndAtomIdx(endIdx);
subMol->addBond(bond,true);
}
}
else {
for(pathIter=path.begin(); pathIter!=path.end(); ++pathIter){
Bond *bond;
bond=mol.getBondWithIdx(*pathIter)->copy();
int begIdx=bond->getBeginAtomIdx();
int endIdx=bond->getEndAtomIdx();
if(atomIdxMap.find(begIdx)==atomIdxMap.end()){
Atom *atom = mol.getAtomWithIdx(begIdx)->copy();
int newAtomIdx=subMol->addAtom(atom,false,true);
atomIdxMap[begIdx] = newAtomIdx;
}
begIdx = atomIdxMap.find(begIdx)->second;
if(atomIdxMap.find(endIdx)==atomIdxMap.end()){
Atom *atom = mol.getAtomWithIdx(endIdx)->copy();
int newAtomIdx=subMol->addAtom(atom,false,true);
atomIdxMap[endIdx] = newAtomIdx;
}
endIdx = atomIdxMap.find(endIdx)->second;
bond->setOwningMol(subMol);
bond->setBeginAtomIdx(begIdx);
bond->setEndAtomIdx(endIdx);
subMol->addBond(bond,true);
}
}
if(mol.getNumConformers()){
// copy coordinates over:
Conformer *conf=new Conformer(subMol->getNumAtoms());
const Conformer &oconf=mol.getConformer();
conf->set3D(oconf.is3D());
for(INT_MAP_INT::const_iterator mapIt=atomIdxMap.begin();
mapIt!=atomIdxMap.end();++mapIt){
conf->setAtomPos(mapIt->second,oconf.getAtomPos(mapIt->first));
}
subMol->addConformer(conf,true);
}
return subMol;
}
PATH_TYPE bondListFromAtomList(const ROMol &mol, const PATH_TYPE &atomIds) {
PATH_TYPE bids;
unsigned int natms = atomIds.size();
if (natms <= 1) {
return bids; //FIX: should probably throw an exception
}
for (unsigned int i = 0; i < natms; i++) {
for (unsigned int j = i+1; j < natms; j++) {
const Bond *bnd = mol.getBondBetweenAtoms(atomIds[i], atomIds[j]);
if (bnd) {
int bid = bnd->getIdx();
bids.push_back(bid);
}
}
}
return bids;
}
using boost::uint32_t;
using boost::int32_t;
DiscrimTuple
calcPathDiscriminators(const ROMol &mol, const PATH_TYPE &path, bool useBO,
std::vector<boost::uint32_t> *extraInvars) {
if(extraInvars) CHECK_INVARIANT(extraInvars->size()==mol.getNumAtoms(),"bad extra invars");
DiscrimTuple res;
// Start by collecting the atoms in the path and their degrees
std::vector<int32_t> atomsUsed(mol.getNumAtoms(),-1); // map from atom index->path index
std::vector<const Atom *> atoms; // to contain the atoms in the path
std::vector<uint32_t> pathDegrees; // degrees of each atom *in the path*
for(PATH_TYPE::const_iterator pathIter=path.begin();
pathIter!=path.end(); ++pathIter){
const Bond *bond=mol.getBondWithIdx(*pathIter);
if(atomsUsed[bond->getBeginAtomIdx()]<0){
atomsUsed[bond->getBeginAtomIdx()]=atoms.size();
atoms.push_back(bond->getBeginAtom());
pathDegrees.push_back(1);
} else {
pathDegrees[atomsUsed[bond->getBeginAtomIdx()]]+=1;
}
if(atomsUsed[bond->getEndAtomIdx()]<0){
atomsUsed[bond->getEndAtomIdx()]=atoms.size();
atoms.push_back(bond->getEndAtom());
pathDegrees.push_back(1);
} else {
pathDegrees[atomsUsed[bond->getEndAtomIdx()]]+=1;
}
}
// Calculate the atomic invariants
unsigned int nAtoms=atoms.size();
std::vector<uint32_t> invars(nAtoms);
for(unsigned int i=0;i<nAtoms;++i){
const Atom *atom=atoms[i];
uint32_t invar=atom->getAtomicNum();
gboost::hash_combine(invar,pathDegrees[i]);
gboost::hash_combine(invar,atom->getFormalCharge());
int deltaMass = static_cast<int>(atom->getMass() -
PeriodicTable::getTable()->getAtomicWeight(atom->getAtomicNum()));
gboost::hash_combine(invar,deltaMass);
if(atom->getIsAromatic()){
gboost::hash_combine(invar,1);
}
if(extraInvars){
gboost::hash_combine(invar,(*extraInvars)[atom->getIdx()]);
}
invars[i] = invar;
}
// now do the Morgan iterations:
// the most number of cycles we need for the atoms on the edges
// to feel each other is pathSize/2
// EFF: it may be worth revisiting this at some point to see
// if the iteration count can be even smaller (and if it
// makes a difference in runtime)
unsigned int nCycles=path.size()/2+1;
gboost::hash<std::vector<uint32_t> > vectHasher;
for(unsigned int cycle=0;cycle<nCycles;++cycle){
// let each atom feel it's neighbors:
std::vector< std::vector<uint32_t> > locInvars(nAtoms);
for(PATH_TYPE::const_iterator pathIter=path.begin();
pathIter!=path.end(); ++pathIter){
const Bond *bond=mol.getBondWithIdx(*pathIter);
uint32_t v1=invars[atomsUsed[bond->getBeginAtomIdx()]];
uint32_t v2=invars[atomsUsed[bond->getEndAtomIdx()]];
if(useBO){
gboost::hash_combine(v1,static_cast<uint32_t>(bond->getBondType()));
gboost::hash_combine(v2,static_cast<uint32_t>(bond->getBondType()));
}
locInvars[atomsUsed[bond->getBeginAtomIdx()]].push_back(v2);
locInvars[atomsUsed[bond->getEndAtomIdx()]].push_back(v1);
}
// we need to sort by the neighbor invariants to be order
// independent:
for(unsigned int i=0;i<nAtoms;++i){
std::sort(locInvars[i].begin(),locInvars[i].end());
invars[i]=vectHasher(locInvars[i]);
}
}
// again, a sort for order independence:
std::sort(invars.begin(),invars.end());
uint32_t pathInvar=vectHasher(invars);
// also include the path size (bond count) and number of atoms
// in the discriminator
return boost::make_tuple(pathInvar,path.size(),nAtoms);
}
//
// This is intended for use on either subgraphs or paths.
// The entries in PATH_LIST should refer to bonds though (not
// atoms)
//
PATH_LIST uniquifyPaths (const ROMol &mol, const PATH_LIST &allPaths,
bool useBO){
PATH_LIST res;
std::vector<DiscrimTuple> discrimsSeen;
for(PATH_LIST::const_iterator path=allPaths.begin();
path!=allPaths.end();++path){
DiscrimTuple discrims = calcPathDiscriminators(mol,*path,useBO);
if(std::find(discrimsSeen.begin(),discrimsSeen.end(),discrims)==discrimsSeen.end()){
discrimsSeen.push_back(discrims);
res.push_back(*path);
}
}
return res;
}
} // end of namespace Subgraphs
} // end of namespace RDKit